性能参数 |
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产品名称 |
HDAC3 Inhibitor |
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规格 |
1mg 5mg 10mg |
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货号 |
GOY-Y3581 |
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含量 |
>98.00% |
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CAS |
2044701-99-5 |
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别名 |
N/A |
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化学名 |
N/A |
分子式 |
C20H23N3O2 |
分子量 |
分子量 337.4 |
溶解度 |
DMF: 10 mg/ml,DMSO: 10 mg/ml,Ethanol: 30 mg/ml |
储存条件 |
Store at -20°C |
General tips |
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用途 |
仅供科研 |
价格 |
电询 |
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详细内容 |
HDAC3 inhibitor is an allosteric inhibitor of histone deacetylase 3 (HDAC3; Ki = 0.16 nM). It is selective for HDAC3 over HDAC1 and HDAC2 (IC50s = 0.95, 11.81, and 95.45 nM, respectively, using recombinant HDACs). In addition, it is selective for acute myeloid, monocytic, and lymphoblastic leukemia cell lines (EC50s = 36.37, 76.64, and 151.7 nM, respectively) over chronic myeloid, acute promyelocytic, and acute lymphoblastic cells (EC50s = 2,160, >10,000, and >10,000 nM, respectively). |
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传真号码:021-39596320 021-39921927
QQ: 3004918891 3004905818 3004901493
移动电话:18321818584 15026555973
地址:上海松江新砖公路1155号
产品均为实验试剂,仅供科研实验使用,非药品、非食品、不可用于动物及人体!