性能参数

产品名称

Stavudine (d4T)

规格

10mM (in 1mL DMSO) 100mg 500mg

货号

GOY-Y3211

 含量

>98.00%

CAS

3056-17-5

别名

化学名

1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]-5-methylpyrimidine-2,4-dione

分子式

C10H12N2O4

分子量

分子量 224.21

溶解度

DMF: 30 mg/ml,DMSO: 30 mg/ml,Ethanol: 10 mg/ml,PBS (pH 7.2): 10 mg/ml

储存条件

Store at -20°C

General tips

用途

仅供科研

价格

电询

详细内容

SB-271046 is a potent, selective and orally active antagonist of 5-HT6 receptor (pKi = 8.9 in HeLa cell in vitro)

5-HT receptor is a G-protein coupled receptor for 5-hydroxytryptamine (serotonin) that found in nerve systems. It also functions as receptor for various alkaloids and psychoactive substances.

In native brain tissue, SB-271046 exhibits high affinity for human recombinant 5-HT6 receptors and 5-HT6 receptors. SB-271046 has a 200 fold greater selectivity over all other 5-HT receptors subtypes tested. [1]

In rat MEST (maximal electroshock seizure threshold) test, SB-271046 increases the seizure threshold over a wide range of dose with a minimum effective dose of 40.1 mg kg71 p.o. and maximum effect at 4 h post-dose. [1] In rat Morris water maze that measuring behavior acquisition and retention, galanthamine and SB-271046 combined treatment reverses the scopolamine- or MK-801-induced learning impairments. [2]

2,4-二甲基-3-吡咯羧酸乙酯  2199-51-1  3,5-二甲基-2-吡咯甲醛  2199-58-8

甲磺酸伊马替尼  220127-57-1  3,4,5-三氟溴苄  220141-72-0

4-羟基-3-三氟甲基苯甲醛  220227-98-5  肉桂酰胺  22031-64-7

吲哚-4-硼酸  220465-43-0  2-乙?；拎? 22047-25-2

FMOC-D-3-(3-噻吩基)-丙氨酸  220497-90-5  5-氟-2-甲基苯甲醛  22062-53-9

1-苄基-4-?

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